Read e-book online Drug Design: Medicinal Chemistry: A Series of Monographs, PDF

By E. J. Ariëns

ISBN-10: 0120603055

ISBN-13: 9780120603053

Drug layout, quantity V covers the elemental techniques to the advance of bioactive compounds. The e-book discusses the usage of operational schemes for analog synthesis in drug layout; the layout of enzyme inhibitors (transition nation analogs); and the importance of structure-absorption-distribution relationships for drug layout.
The textual content describes the function of charge-transfer approaches within the motion of bioactive fabrics, in addition to the techniques to the rational mixture of antimetabolites for melanoma chemotherapy. The physicochemical, quantum chemical, and different theoretical recommendations for the knowledge of the mechanism of motion of relevant apprehensive procedure (CNS) brokers, corresponding to psychoactive medicines, narcotics, and narcotic antagonists and anesthetics, also are encompassed.
Chemists, biochemists, pharmacologists, and other people occupied with drug layout will locate the ebook invaluable.

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Read Online or Download Drug Design: Medicinal Chemistry: A Series of Monographs, Vol. 5 PDF

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Drug Design: Medicinal Chemistry: A Series of Monographs, Vol. 5 by E. J. Ariëns

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